MICHÈLE REBOUD-RAVAUX: шукати на сайті Z-Library

Lucia Formicola, Xavier Maréchal, Nicolas Basse, Michelle Bouvier-Durand, Danièle Bonnet-Delpon, Thierry Milcent, Michèle Reboud-Ravaux, Sandrine Ongeri

Рік:

2006

Мова:

english

Файл:

PDF, 197 KB

english, 2006

Novel fluorinated pseudopeptides as proteasome inhibitors

Журнал:

Florence Lebon, Eve de Rosny, Michèle Reboud-Ravaux, François Durant

Рік:

2009

Мова:

english

Файл:

PDF, 172 KB

english, 2009

De novo drug design of a new copper chelate molecule acting as HIV-1 protease inhibitor

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

1998

Мова:

english

Файл:

PDF, 380 KB

english, 1998

Inhibition of human leukocyte elastase by functionalized N-aryl-3,3-dihalogenoazetidin-2-ones. Stereospecific synthesis and chiral recognition of dissymmetrically C3-substituted β-lactams

Caroline Doucet, Isabelle Vergely, Michèle Reboud-Ravaux, Jean Guilhem, Randa Kobaiter, Roger Joyeau, Michel Wakselman

Журнал:

Tetrahedron: Asymmetry

Рік:

1997

Мова:

english

Файл:

PDF, 840 KB

english, 1997

Coumarinic derivatives as mechanism-based inhibitors of α-chymotrypsin and human leukocyte elastase

Lionel Pochet, Caroline Doucet, Georges Dive, Johan Wouters, Bernard Masereel, Michèle Reboud-Ravaux, Bernard Pirotte

Журнал:

Рік:

2000

Мова:

english

Файл:

PDF, 390 KB

english, 2000

Synthesis of N-glyoxylyl peptides and their in vitro evaluation as HIV-1 protease inhibitors

Driss Qasmi, Eve de Rosny, Loïc René, Bernard Badet, Isabelle Vergely, Nicole Boggetto, Michèle Reboud-Ravaux

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

1997

Мова:

english

Файл:

PDF, 650 KB

english, 1997

Synthesis and activity of HIV protease inhibitors

Patrick Garrouste, Macek Pawlowski, Thierry Tonnaire, Sames Sicsic, Pascal Dumy, Eve de Rosny, Michèle Reboud-Ravaux, Pierre Fulcrand, Jean Martinez

Журнал:

Guy, Laure, Vidal, Joëlle, Collet, André, Amour, Augustin, Reboud-Ravaux, Michèle

Рік:

1998

Мова:

english

Файл:

PDF, 1.01 MB

english, 1998

Design and Synthesis of Hydrazinopeptides and Their Evaluation as Human Leukocyte Elastase Inhibitors

Журнал:

Basse, Nicolas, Montes, Matthieu, Maréchal, Xavier, Qin, Lixian, Bouvier-Durand, Michelle, Genin, Emilie, Vidal, Joëlle, Villoutreix, Bruno O., Reboud-Ravaux, Michèle

Рік:

1998

Мова:

english

Файл:

PDF, 197 KB

english, 1998

Novel Organic Proteasome Inhibitors Identified by Virtual and in Vitro Screening

Журнал:

Michéle Reboud-Ravaux, Giséle Desvages

Рік:

2010

Мова:

english

Файл:

PDF, 793 KB

english, 2010

Inactivation of human high- and low-molecular-weight urokinases: Analysis of their active site

Журнал:

Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology

Рік:

1984

Мова:

english

Файл:

PDF, 762 KB

english, 1984

Reaction of thrombin and proteinases of the fibrinolytic system with a mechanism-based inhibitor, 3,4-dihydro-3-benzyl-6-chloromethylcoumarin

Amram Mor, Jean Maillard, Catherine Favreau, Michèle Reboud-Ravaux

Журнал:

Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology

Рік:

1990

Мова:

english

Файл:

PDF, 527 KB

english, 1990

Acyloxybenzyl halides, inhibitors of elastases

Anne-Cécile Vilain, Veronica Okochi, Isabelle Vergely, Michèle Reboud-Ravaux, Jean-Paul Mazaleyrat, Michel Wakselman

Журнал:

Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology

Рік:

1991

Мова:

english

Файл:

PDF, 374 KB

english, 1991

A new series of N5 derivatives of the 1,1,5-trimethyl furo[3,4-c]pyridine-3,4-dione (cerpegin) selectively inhibits the post-acid activity of mammalian 20S proteasomes

The Hien Pham, Anna Hovhannisyan, Dominique Bouvier, Lei Tian, Michèle Reboud-Ravaux, Gagik Melikyan, Michelle Bouvier-Durand

Журнал:

Рік:

2012

Мова:

english

Файл:

PDF, 1.17 MB

english, 2012

Noncovalent inhibition of 20S proteasome by pegylated dimerized inhibitors

Xavier Maréchal, Anaïs Pujol, Nicolas Richy, Emilie Genin, Nicolas Basse, Michèle Reboud-Ravaux, Joëlle Vidal

Журнал:

Julien Dumond, Nicole Boggetto, Hans J. Schramm, Wolfgang Schramm, Masayuki Takahashi, Michèle Reboud-Ravaux

Рік:

2012

Мова:

english

Файл:

PDF, 440 KB

english, 2012

Metal-organic compounds: a new approach for drug discovery: N1-(4-methyl-2-pyridyl)-2,3,6-trimethoxybenzamide copper(II) complex as an inhibitor of human immunodeficiency virus 1 protease

Florence Lebon, Nicole Boggetto, Marie Ledecq, François Durant, Zohra Benatallah, Sames Sicsic, René Lapouyade, Olivier Kahn, Ange Mouithys-Mickalad, Ginette Deby-Dupont, Michèle Reboud-Ravaux

Журнал:

Biochemical Pharmacology

Рік:

2002

Мова:

english

Файл:

PDF, 409 KB

english, 2002

Thyroxine-derivatives of lipopeptides: bifunctional dimerization inhibitors of human immunodeficiency virus-1 protease

Журнал:

Biochemical Pharmacology

Рік:

2003

Мова:

english

Файл:

PDF, 230 KB

english, 2003

Synthesis and enzymic hydrolysis of cyclic peptides containing an anthranilic acid residue

JEAN-PAUL MAZALEYRAT, MICHÈLE REBOUD-RAVAUX, MICHEL WAKSELMAN

Журнал:

Chemical Biology & Drug Design

Рік:

1987

Мова:

english

Файл:

PDF, 868 KB

english, 1987

Synthesis and protease-catalyzed hydrolysis of a novel hydrazinopeptide

AUGUSTIN AMOUR, ANDRÉ COLLET, CATHERINE DUBAR, MICHÈLE REBOUD-RAVAUX

Журнал:

Chemical Biology & Drug Design

Рік:

1994

Мова:

english

Файл:

PDF, 750 KB

english, 1994

N-Acetylbenzotriazole as a Protein Reagent : Specific Behaviour towards δ-Chymotrypsin

Michèle REBOUD-RAVAUX, Charis GHELIS

Журнал:

FEBS Journal

Рік:

1976

Мова:

english

Файл:

PDF, 802 KB

english, 1976

ChemInform Abstract: A New Series of N5 Derivatives of the 1,1,5-Trimethyl Furo[3,4-c]pyridine-3,4-dione (Cerpegin) Selectively Inhibits the Post-Acid Activity of Mammalian 20S Proteasomes.

The Hien Pham, Anna Hovhannisyan, Dominique Bouvier, Lei Tian, Michele Reboud-Ravaux, Gagik Melikyan, Michelle Bouvier-Durand

Журнал:

ChemInform

Рік:

2012

Файл:

PDF, 27 KB

2012

A cyclopeptidic suicide substrate preferentially inactivates urokinase-type plasminogen activator

Michèle Reboud-Ravaux, Anne-Cécile Vilain, Nicole Boggetto, Jean Maillard, Catherine Favreau, Juan Xie, Jean-Paul Mazaleyrat, Michel Wakselman

Журнал:

Biochemical and Biophysical Research Communications

Рік:

1991

Мова:

english

Файл:

PDF, 524 KB

english, 1991

Protection of vascular basement membrane and microcirculation from elastase-induced damage with a fluorinated β-lactam derivative

Jean-Louis Maillard, Catherine Favreau, Isabelle Vergely, Michèle Reboud-Ravaux, Roger Joyeau, Randa Kobaiter, Michel Wakselman

Журнал:

Clinica Chimica Acta

Рік:

1992

Мова:

english

Файл:

PDF, 901 KB

english, 1992

Role of monocyte/macrophage derived matrix-metalloproteinases (gelatinases) in prolonged skin inflammation

Jean L. Maillard, Catherine Favreau, Michèle Reboud-Ravaux

Журнал:

Clinica Chimica Acta

Рік:

1995

Мова:

english

Файл:

PDF, 934 KB

english, 1995

Functionalized N-aryl azetidinones as novel mechanism-based inhibitors of neutrophil elastase

Michel Wakselman, Roger Joyeau, Randa Kobaiter, Nicole Boggetto, Isabelle Vergely, Jean Maillard, Veronica Okochi, Jean-Jacques Montagne, Michèle Reboud-Ravaux

Журнал:

FEBS Letters

Рік:

1991

Мова:

english

Файл:

PDF, 574 KB

english, 1991

Liberation of an N-terminal proline-rich peptide from the cryptic proteinase of fibronectin by auto-proteolysis

Maurice Pagano, Gilles Clodic, Gérard Bolbach, Magalie Michiel, Saliha Haddag, Michèle Reboud-Ravaux

Журнал:

Archives of Biochemistry and Biophysics

Рік:

2008

Мова:

english

Файл:

PDF, 828 KB

english, 2008

Towards the control of intracellular protein turnover: Mitochondrial Lon protease inhibitors versus proteasome inhibitors

Aurélien Bayot, Nicolas Basse, Irene Lee, Monique Gareil, Bernard Pirotte, Anne-Laure Bulteau, Bertrand Friguet, Michèle Reboud-Ravaux

Журнал:

Biochimie

Рік:

2008

Мова:

english

Файл:

PDF, 347 KB

english, 2008

Coumarinic derivatives show anti-inflammatory effects on alveolar macrophages, but their anti-elastase activity is essential to reduce lung inflammation in vivo

Elyse Y. Bissonnette, Guy M. Tremblay, Véronique Turmel, Bernard Pirotte, Michèle Reboud-Ravaux

Журнал:

International Immunopharmacology

Рік:

2009

Мова:

english

Файл:

PDF, 513 KB

english, 2009

Regulation of the 26S proteasome activities by peptides mimicking cleavage products

David Papapostolou, Olivier Coux, Michèle Reboud-Ravaux

Журнал:

Biochemical and Biophysical Research Communications

Рік:

2002

Мова:

english

Файл:

PDF, 169 KB

english, 2002

Stereoselective Synthesis of Peptidyl Trifluoromethyl Alcohols and Ketones: Inhibitory Potency Against Human Leucocyte Elastase, Cathepsin G, Porcine Pancreatic Elastase and HIV-1 Protease

AUGUSTIN AMOUR, MICHÈLE REBOUD-RAVAUX, EVE DE ROSNY, AHMED ABOUABDELLAH, JEAN-PIERRE BÉGUÉ, DANIÈLE BONNET-DELPON, MARIE LE GALL

Журнал:

Journal of Pharmacy and Pharmacology

Рік:

1998

Мова:

english

Файл:

PDF, 712 KB

english, 1998

Dimerized Linear Mimics of a Natural Cyclopeptide (TMC-95A) Are Potent Noncovalent Inhibitors of the Eukaryotic 20S Proteasome

Desvergne, Audrey, Genin, Emilie, Maréchal, Xavier, Gallastegui, Nerea, Dufau, Laure, Richy, Nicolas, Groll, Michael, Vidal, Joëlle, Reboud-Ravaux, Michèle

Журнал:

Bannwarth, Ludovic, Kessler, Albane, Pèthe, Stéphanie, Collinet, Bruno, Merabet, Naïma, Boggetto, Nicole, Sicsic, Sames, Reboud-Ravaux, Michèle, Ongeri, Sandrine

Рік:

2013

Мова:

english

Файл:

PDF, 1.37 MB

english, 2013

Molecular Tongs Containing Amino Acid Mimetic Fragments: New Inhibitors of Wild-Type and Mutated HIV-1 Protease Dimerization

Журнал:

Рік:

2006

Мова:

english

Файл:

PDF, 173 KB

english, 2006

Esters and Amides of 6-(Chloromethyl)-2-oxo-2 H -1-benzopyran-3-carboxylic Acid as Inhibitors of α-Chymotrypsin: Significance of the “Aromatic” Nature of the Novel Ester-Type Coumarin for Strong Inhibitory Activity

Pochet, Lionel, Doucet, Caroline, Schynts, Marc, Thierry, Nicole, Boggetto, Nicole, Pirotte, Bernard, Jiang, Kai Y., Masereel, Bernard, de Tullio, Pascal, Delarge, Jacques, Reboud-Ravaux, Michèle

Журнал:

Tan, Xiao, Furio, Laetitia, Reboud-Ravaux, Michèle, Villoutreix, Bruno O., Hovnanian, Alain, El Amri, Chahrazade

Рік:

1996

Мова:

english

Файл:

PDF, 193 KB

english, 1996

1,2,4-Triazole derivatives as transient inactivators of kallikreins involved in skin diseases

Журнал:

Doucet, Caroline, Pochet, Lionel, Thierry, Nicole, Pirotte, Bernard, Delarge, Jacques, Reboud-Ravaux, Michèle

Рік:

2013

Мова:

english

Файл:

PDF, 945 KB

english, 2013

6-Substituted 2-Oxo-2 H -1-benzopyran-3-carboxylic Acid as a Core Structure for Specific Inhibitors of Human Leukocyte Elastase †

Журнал:

Sebastien Lyonnais,Laure Dufau,Michele Reboud-Ravaux,Roland Marquet…

Рік:

1999

Мова:

english

Файл:

PDF, 228 KB

english, 1999

RNA remarkably promotes HIV-1 protease fast turnover for NCp15 processing in mild acidic conditions leading to condensation of HIV-1 nucleocapsid

Журнал:

Retrovirology

Рік:

2013

Мова:

english

Файл:

PDF, 76 KB

english, 2013

New C4- and C1-derivatives of furo[3,4-c]pyridine-3-ones and related compounds: Evidence for site-specific inhibition of the constitutive proteasome and its immunoisoform

Hovhannisyan, Anna, Pham, The Hien, Bouvier, Dominique, Piroyan, Alexander, Dufau, Laure, Qin, Lixian, Cheng, Yan, Melikyan, Gagik, Reboud-Ravaux, Michèle, Bouvier-Durand, Michelle

Журнал:

Hovhannisyan, Anna, Pham, The Hien, Bouvier, Dominique, Qin, Lixian, Melikyan, Gagik, Reboud-Ravaux, Michèle, Bouvier-Durand, Michelle

Рік:

2014

Мова:

english

Файл:

PDF, 6.63 MB

english, 2014

Les activateurs du plasminogène: aspects généraux et développements récents

Reboud-Ravaux, Michèle

Журнал:

Biochimie

Рік:

1985

Файл:

PDF, 1.70 MB

1985

C1 and N5 derivatives of cerpegin: Synthesis of a new series based on structure–activity relationships to optimize their inhibitory effect on 20S proteasome

Журнал:

Tan, Xiao, Bertonati, Claudia, Qin, Lixian, Furio, Laetitia, El Amri, Chahrazade, Hovnanian, Alain, Reboud-Ravaux, Michèle, Villoutreix, Bruno O.

Рік:

2013

Мова:

english

Файл:

PDF, 917 KB

english, 2013

Identification by in silico and in vitro screenings of small organic molecules acting as reversible inhibitors of kallikreins

Журнал:

Bouras, Ahmed, Boggetto, Nicole, Benatalah, Zohra, de Rosny, Eve, Sicsic, Sames, Reboud-Ravaux, Michèle

Рік:

2013

Мова:

english

Файл:

PDF, 1.25 MB

english, 2013

Design, Synthesis, and Evaluation of Conformationally Constrained Tongs, New Inhibitors of HIV-1 Protease Dimerization

Журнал:

Basse, Nicolas, Piguel, Sandrine, Papapostolou, David, Ferrier-Berthelot, Alexandra, Richy, Nicolas, Pagano, Maurice, Sarthou, Pierre, Sobczak-Thépot, Joëlle, Reboud-Ravaux, Michèle, Vidal, Joëlle

Рік:

1999

Мова:

english

Файл:

PDF, 162 KB

english, 1999

Linear TMC-95-Based Proteasome Inhibitors

Журнал:

Altei, Wanessa F., Picchi, Douglas G., Abissi, Barbara M., Giesel, Guilherme M., Flausino, Otavio, Reboud-Ravaux, Michèle, Verli, Hugo, Crusca, Edson, Silveira, Edilberto R., Cilli, Eduardo M., Bolzan

Рік:

2007

Мова:

english

Файл:

PDF, 168 KB

english, 2007

Jatrophidin I, a cyclic peptide from Brazilian Jatropha curcas L.: Isolation, characterization, conformational studies and biological activity

Журнал:

Phytochemistry

Рік:

2014

Мова:

english

Файл:

PDF, 756 KB

english, 2014

New mechanism-based inactivators of trypsin-like proteinases. Selective inactivation of urokinase by functionalized cyclopeptides incorporating a sulfoniomethyl-substituted m-aminobenzoic acid residue

Wakselman, Michel, Xie, Juan, Mazaleyrat, Jean Paul, Boggetto, Nicole, Vilain, Anne Cecile, Montagne, Jean Jacques, Reboud-Ravaux, Michele

Журнал:

Merabet, Naïma, Dumond, Julien, Collinet, Bruno, Van Baelinghem, Laurence, Boggetto, Nicole, Ongeri, Sandrine, Ressad, Fariza, Reboud-Ravaux, Michèle, Sicsic, Sames

Рік:

1993

Мова:

english

Файл:

PDF, 1.12 MB

english, 1993

New Constrained “Molecular Tongs” Designed To Dissociate HIV-1 Protease Dimer

Журнал: